High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists
Raphaël Bolteau, Romain Duroux, Amélie Laversin, Brandon Vreulz, Anna Shiriaeva, Benjamin Stauch, Gye Won Han, Vadim Cherezov, Nicolas Renault, Amélie Barczyk, Séverine Ravez, Mathilde Coevoet, Patricia Melnyk, Maxime Liberelle, Saı̈d Yous
Topics & Concepts
Adenosine receptorChemistryAntagonistLigand (biochemistry)AdenosineQuinazolineReceptorStereochemistryDocking (animal)PharmacologyCombinatorial chemistryBiochemistryMedicineAgonistNursingAdenosine and Purinergic SignalingPharmacological Receptor Mechanisms and EffectsReceptor Mechanisms and Signaling