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Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives

Endika Martín‐Encinas, Asier Selas, Cinzia Tesauro, Gloria Rubiales, Birgitta R. Knudsen, Francisco Palácios, Concepción Alonso

2020European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryStereochemistryTopoisomeraseEnzymeOrganic chemistryCancer therapeutics and mechanismsSynthesis and Biological ActivitySynthesis and Biological Evaluation
Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives | Litcius