Development of a sensitive luminescent probe to uncover new BRD4 inhibitors in living cells
Yingqi Song, Ke‐Jia Wu, Zhiming Zhang, Tzu‐Ming Liu, Chung-Nga Ko, Wei-Guo Zhu, Dik‐Lung Ma, Wanhe Wang, Chung‐Hang Leung
Topics & Concepts
BRD4ChemistryBiophysicsCytoplasmCancer cellBromodomainHistoneCancer researchBiochemistryCancerBiologyGeneticsDNAProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsHistone Deacetylase Inhibitors Research