Litcius/Paper detail

Structural modification aimed for improving solubility of lead compounds in early phase drug discovery

Bhanuranjan Das, Anurag T. K. Baidya, Alen T. Mathew, Ashok Kumar Yadav, Rajnish Kumar

2022Bioorganic & Medicinal Chemistry171 citationsDOIOpen Access PDF

Topics & Concepts

SolubilityChemistryDrug discoveryBioavailabilityCombinatorial chemistryDrugProdrugDrug developmentOrganic chemistryBiochemical engineeringPharmacologyBiochemistryMedicineEngineeringComputational Drug Discovery MethodsCrystallization and Solubility StudiesPhenothiazines and Benzothiazines Synthesis and Activities