Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors
Maria Giulia Nizi, Jenny Desantis, Yoshio Nakatani, Serena Massari, Maria Angela Mazzarella, Gauri Shetye, Stefano Sabatini, Maria Letizia Barreca, Giuseppe Manfroni, Tommaso Felicetti, Rowena Rushton-Green, Kiel Hards, Gniewomir Latacz, Grzegorz Satała, Andrzej J. Bojarski, Violetta Cecchetti, Michal H. Kolář, Jadwiga Handzlik, Gregory M. Cook, Scott G. Franzblau, Oriana Tabarrini
Topics & Concepts
ChemistryLead compoundBedaquilineMycobacterium tuberculosisCombinatorial chemistryEnzymeOxidoreductaseBiochemistryStereochemistryPharmacologyTuberculosisIn vitroMedicinePathologyPhenothiazines and Benzothiazines Synthesis and ActivitiesChemical Reaction MechanismsCancer therapeutics and mechanisms