Selectively targeting individual bromodomain: Drug discovery and molecular mechanisms
Qianqian Wang, Xiaomin Shao, Elaine Lai Han Leung, Yingqing Chen, Xiaojun Yao
Topics & Concepts
BromodomainDrug discoveryComputational biologyBRD4DrugProteolysisChemistryBiologyPharmacologyBioinformaticsEpigeneticsBiochemistryEnzymeGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsPeptidase Inhibition and Analysis