Design, synthesis, and pharmacological evaluation of indole-piperidine amides as Blood−brain barrier permeable dual cholinesterase and β-secretase inhibitors
Razia Banoo, Vijay K. Nuthakki, Bhagyashri N. Wadje, Ankita Sharma, Sandip B. Bharate
Topics & Concepts
ChemistryPiperidineIndole testBlood–brain barrierCholinesteraseCarboxamidePharmacologyStereochemistryCombinatorial chemistryBiochemistryCentral nervous systemNeuroscienceBiologyMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsNicotinic Acetylcholine Receptors Study