Ketamine and Major Ketamine Metabolites Function as Allosteric Modulators of Opioid Receptors
Ivone Gomes, Achla Gupta, Elyssa B. Margolis, Lloyd D. Fricker, Lakshmi A. Devi
Topics & Concepts
PharmacologyKetamineChemistryOpioidReceptorEnkephalinAllosteric modulatorAgonistDynorphinNMDA receptorDAMGOGlutamate receptorAllosteric regulationNaltrexoneκ-opioid receptorOpioid peptideBiologyBiochemistryNeuroscienceTreatment of Major DepressionNeuroscience and Neuropharmacology ResearchReceptor Mechanisms and Signaling