Copper-mediated radioiodination and radiobromination via aryl boronic precursor and its application to 125I/77Br–labeled prostate-specific membrane antigen imaging probes
Yuto Kondo, Hiroyuki Kimura, Ichiro Sasaki, Shigeki Watanabe, Yasuhiro Ohshima, Yusuke Yagi, Yasunao Hattori, Manami Koda, Hidekazu Kawashima, Hiroyuki Yasui, Noriko S. Ishioka
Topics & Concepts
ChemistryPeptidomimeticRadiosynthesisCombinatorial chemistryBioorthogonal chemistryBiodistributionImaging agentPharmacophoreArylChemical synthesisPeptideStereochemistryBiochemistryOrganic chemistryClick chemistryIn vivoBiotechnologyAlkylIn vitroBiologyRadiopharmaceutical Chemistry and ApplicationsPeptidase Inhibition and AnalysisProstate Cancer Treatment and Research