Design, synthesis, and biological evaluation of 4-(2-fluorophenoxy)-7-methoxyquinazoline derivatives as dual EGFR/c-Met inhibitors for the treatment of NSCLC
Sheng Tang, Chuanchuan Sun, Xintao He, Wenhui Gan, Linxiao Wang, Dan Qiao, Xinyu Guan, Shan Xu, Pengwu Zheng, Wufu Zhu
Topics & Concepts
ChemistryEpidermal growth factor receptorA549 cellApoptosisEGFR inhibitorsPharmacologyProtein kinase BAfatinibIn vivoCell cycle checkpointCell growthCell cycleC-MetCancer researchReceptorErlotinibBiochemistryHepatocyte growth factorBiologyBiotechnologyLung Cancer Treatments and MutationsHER2/EGFR in Cancer ResearchPeptidase Inhibition and Analysis