Chemical proteomic profiling with photoaffinity labeling strategy identifies antimalarial targets of artemisinin
Peng Gao, Jiayun Chen, Peng Sun, Jianyou Wang, Jianyou Wang, Huan Tang, Fei Xia, Liwei Gu, Huimin Zhang, Chen Wang, Yin Kwan Wong, Yinhua Zhu, Chengchao Xu, Chengchao Xu, Jigang Wang, Jigang Wang
Topics & Concepts
ArtemisininPhotoaffinity labelingChemistryCovalent bondAntimalarial AgentCovalent bindingPlasmodium falciparumCombinatorial chemistryChemical biologyDrug discoveryComputational biologyBiochemistryMalariaBinding siteBiologyOrganic chemistryImmunologyMalaria Research and ControlComputational Drug Discovery MethodsHIV/AIDS drug development and treatment