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Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors

Vladlen Klochkov, Elena N. Bezsonova, Meriam Dubar, Daria D. Melekhina, Victor V. Temnov, Ekaterina V. Zaryanova, Natalia A. Lozinskaya, Denis A. Babkov, А. А. Спасов

2021Bioorganic & Medicinal Chemistry Letters17 citationsDOIOpen Access PDF

Topics & Concepts

PostprandialChemistryIn vivoAcarbosePharmacologyIn vitroDiabetes mellitusPotencyBiochemistryEnzymeEndocrinologyMedicineBiologyBiotechnologyNatural Antidiabetic Agents StudiesPhytochemicals and Antioxidant ActivitiesAdvanced Glycation End Products research
Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors | Litcius