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Structural basis for CaVα2δ:gabapentin binding

Zhou Chen, Abhisek Mondal, Daniel L. Minor

2023Nature Structural & Molecular Biology39 citationsDOIOpen Access PDF

Topics & Concepts

GabapentinGene isoformChemistryCalcium channelSelectivityBinding siteBiophysicsGeneCalciumBiochemistryBiologyMedicinePathologyCatalysisOrganic chemistryAlternative medicineIon channel regulation and functionCardiac electrophysiology and arrhythmiasReceptor Mechanisms and Signaling
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