Structural mechanism underlying ligand binding and activation of PPARγ
Jinsai Shang, Douglas J. Kojetin
Topics & Concepts
Isothermal titration calorimetryLigand (biochemistry)ChemistryAllosteric regulationSurface plasmon resonanceAgonistBiophysicsBinding siteNuclear receptorStereochemistryConformational changePlasma protein bindingReceptorBiochemistryBiologyNanotechnologyMaterials scienceNanoparticleTranscription factorGenePeroxisome Proliferator-Activated ReceptorsDrug Transport and Resistance MechanismsMetabolism, Diabetes, and Cancer