Effect of Conjugation Site and Technique on the Stability and Pharmacokinetics of Antibody-Drug Conjugates
Anna Kaempffe, Stephan Dickgießer, Nicolas Rasche, Andrea Paoletti, Elisa Bertotti, Ilse De Salve, Federico Riccardi Sirtori, Roland Kellner, Doreen Könning, Stefan Hecht, Jan Anderl, Harald Kolmar, Christian Schröter
Topics & Concepts
ConjugateChemistryCysteineMonoclonal antibodyAntibodyConjugated systemIn vivoPharmacokineticsIn vitroAntibody-drug conjugateBiochemistryEnzymePharmacologyBiologyImmunologyBiotechnologyMathematicsPolymerOrganic chemistryMathematical analysisHER2/EGFR in Cancer ResearchMonoclonal and Polyclonal Antibodies ResearchBiosimilars and Bioanalytical Methods