Prediction of drug-drug interaction risk of P-glycoprotein substrate in drug discovery
Yasuto Kido, Isamu Nanchi, Takanobu Matsuzaki, Ryosuke Watari, Hayato Kiyohara, Naomi M. Seki, Tomohiko Okuda
Topics & Concepts
P-glycoproteinPharmacokineticsDrugPharmacologyArea under the curveDrug-drug interactionEffluxChemistryInternal medicineMedicineBiochemistryMultiple drug resistanceAntibioticsDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesPharmacogenetics and Drug Metabolism