Structure, function and pharmacology of human itch GPCRs
Can Cao, Hye Jin Kang, Isha Singh, He Chen, Chengwei Zhang, Wenlei Ye, Byron W. Hayes, Jing Liu, Ryan H. Gumpper, Brian J. Bender, Samuel T. Slocum, B. Krumm, Katherine Lansu, John D. McCorvy, Wesley K. Kroeze, Justin G. English, Jeffrey F. DiBerto, Reid H. J. Olsen, Xi‐Ping Huang, Shicheng Zhang, Yongfeng Liu, Kuglae Kim, Joel Karpiak, Lily Yeh Jan, Soman N. Abraham, Jian Jin, Brian K. Shoichet, Jonathan F. Fay, Bryan L. Roth
Topics & Concepts
G protein-coupled receptorAgonistReceptorAntagonistMast cellEndogenous agonistPharmacologyEndogenyCell biologyChemistryBiologyBiochemistryImmunologyDopamine receptor D1Receptor Mechanisms and SignalingAsthma and respiratory diseasesMast cells and histamine