Does targeting Arg98 of FimH lead to high affinity antagonists?
Tihomir Tomašič, Said Rabbani, Roman P. Jakob, Andreas Reisner, Žiga Jakopin, Timm Maier, Beat Ernst, Marko Anderluh
Topics & Concepts
ChemistryMoietyFimbriaLead compoundLectinBinding affinitiesStereochemistryCarboxylic acidAffinitiesCombinatorial chemistryMutantBinding siteEscherichia coliBiochemistryMicrobiologyReceptorIn vitroBiologyGeneEscherichia coli research studiesAntibiotic Resistance in BacteriaDrug Transport and Resistance Mechanisms