Discovery of novel hydroxyamidine based indoleamine 2,3-dioxygenase 1 (IDO1) and thioredoxin reductase 1 (TrxR1) dual inhibitors
Ji Zhou, Lizhen Yu, Yali Fan, Ci-Hao Guo, Xiaomei Lv, Zhiyin Zhou, Huidan Huang, Dong‐Dong Miao, Shengpeng Zhang, Xinyu Li, Pingping Zhao, Xiaoping Liu, Weihua Hu, Chao Zhang
Topics & Concepts
Indoleamine 2,3-dioxygenaseChemistryKynurenineThioredoxin reductaseIn vivoApoptosisPharmacologyCancer researchThioredoxinIC50BiochemistryIn vitroEnzymeBiologyTryptophanBiotechnologyAmino acidTryptophan and brain disordersPharmacological Receptor Mechanisms and EffectsImmune cells in cancer