Design, synthesis, and characterization of novel aminoalcohol quinolines with strong in vitro antimalarial activity
Alexandra Dassonville‐Klimpt, Jérémy Schneider, Céline Damiani, Camille Tisnerat, Anita Cohen, Nadine Azas, Mathieu Marchivie, Jean Guillon, Catherine Mullié, Patrice Agnamey, Anne Totet, Jérôme Dormoi, Nicolas Taudon, Bruno Pradines, Pascal Sonnet
Topics & Concepts
ChemistryPlasmodium bergheiSelectivityIn vivoIn vitroPlasmodium falciparumIC50StereochemistryMalariaPharmacologyCombinatorial chemistryBiochemistryBiologyImmunologyBiotechnologyCatalysisMalaria Research and ControlComputational Drug Discovery MethodsHIV/AIDS drug development and treatment