Comprehensive analysis of resorcinyl-imidazole Hsp90 inhibitor design
Marius Gedgaudas, Paulina Kaziukonytė, Visvaldas Kairys, Aurelija Mickevičiu̅tė, Asta Zubrienė, A. Brukstus, Daumantas Matulis, Egidijus Kazlauskas
Topics & Concepts
ChemistryImidazoleHsp90 inhibitorHsp90StereochemistryPharmacologyCombinatorial chemistryBiochemistryHeat shock proteinMedicineGeneHeat shock proteins researchComputational Drug Discovery MethodsProtein Structure and Dynamics