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The Metabolism and Disposition of Brepocitinib in Humans and Characterization of the Formation Mechanism of an Aminopyridine Metabolite

Martin E. Dowty, Ruolun Qiu, Alyssa Dantonio, Mark Niosi, Angela C. Doran, Amanda Balesano, Stephen W. Wright, Gregory S. Walker, Raman Sharma

2024Drug Metabolism and Disposition10 citationsDOIOpen Access PDF

Topics & Concepts

DispositionMetaboliteMechanism (biology)4-AminopyridineMetabolismChemistryPharmacologyBiochemistryBiologyPsychologyPhilosophyEndocrinologyPotassium channelEpistemologySocial psychologyChronic Lymphocytic Leukemia ResearchChronic Myeloid Leukemia TreatmentsAcute Lymphoblastic Leukemia research