Elucidating pathway-selective biased CCKBR agonism for Alzheimer’s disease treatment
Jiale Wang, Xue-Ying Sha, Yue Shao, Zi-Hao Zhang, Shen-Ming Huang, Hui Lin, Shiyi Gan, Nan Zhang, Xinyi Xia, Yunan Sun, Jin-Hui Ding, Ruiqi Zhao, Jie Cheng, Pan Shang, Jinpeng Wang, Yanjun Liu, Fan Yang, Peng Xiao, Lu-Wen Wang, Dongyu Zhao, Yi Tang, Lu Tie, Yang Du, Yong E. Zhang, Jufang He, Jin‐Peng Sun
Topics & Concepts
AgonistBiologyCholecystokinin B receptorCholecystokininReceptorNeuroscienceSignal transductionFunctional selectivityDownregulation and upregulationLong-term potentiationEntorhinal cortexEndogenyCholecystokinin receptorInternal medicineG protein-coupled receptorPharmacologyEndocrinologyDiseasePartial agonistCell biologyAnisomycinNeuropeptides and Animal PhysiologyAlzheimer's disease research and treatmentsReceptor Mechanisms and Signaling