Annual review of PROTAC degraders as anticancer agents in 2022
Xiao Wang, Zhao-Long Qin, Na Li, Mei-Qi Jia, Qiu-Ge Liu, Yi‐Ru Bai, Jian Song, Shuo Yuan, Sai‐Yang Zhang
Topics & Concepts
ChemistryPharmacologyMedicineProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisUbiquitin and proteasome pathways