New biologically dynamic hybrid pharmacophore triazinoindole-based-thiadiazole as potent α-glucosidase inhibitors: In vitro and in silico study
Aftab Ahmad Khan, Fazal Rahim, Muhammad Taha, Wajid Rehman, Naveed Iqbal, Abdul Wadood, Nisar Ahmad, Syed Adnan Alı Shah, Mohammed M. Ghoneim, Sultan Alshehri, Mohammed Salahuddin, Khalid Mohammed Khan
Topics & Concepts
AcarbosePharmacophoreChemistryStereochemistryIC50Docking (animal)In silicoIn vitroActive compoundBiological activityEnzymeBiochemistryGeneMedicineNursingSynthesis and biological activitySynthesis and Characterization of Heterocyclic CompoundsClick Chemistry and Applications