Litcius/Paper detail

Design, synthesis and antitumor activity of novel thiophene- triazine derivatives bearing arylurea unit as potent PI3K/mTOR inhibitorss

Shan Xu, Leixuan Luo, Xin Sun, Yang Yang, Qiuyan Guo, Zhiyan Jiang, Yingliang Wu

2022Bioorganic & Medicinal Chemistry23 citationsDOIOpen Access PDF

Topics & Concepts

HeLaPI3K/AKT/mTOR pathwayChemistryKinaseCell cultureCytotoxicityIC50Cancer cellPharmacologyCancerStereochemistryCellBiochemistryIn vitroSignal transductionBiologyGeneticsSynthesis and Characterization of Heterocyclic CompoundsSynthesis and biological activityCancer Mechanisms and Therapy