Synthesis, intramolecular cyclization, and antinociceptive activity of 4-(het)aryl-2-{[4-(4-chlorophenyl)-3-(ethoxycarbonyl)thiophen-2-yl]amino}-4-oxobut-2-enoic acids
I. A. Gorbunova, I. P. Nikonov, Р. Р. Махмудов, D. A. Shipilovskikh, P. S. Silaichev, Sergei A. Shipilovskikh
Topics & Concepts
ChemistryIntramolecular forceThiopheneArylStereochemistryMedicinal chemistryOrganic chemistryAlkylChemical synthesis and pharmacological studiesSynthesis and Characterization of PyrrolesSynthesis and Reactivity of Heterocycles