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Preclinical evaluation of chemically reactive metabolites and mitigation of bioactivation in drug discovery

Chunyong He, Yuchang Mao, Hong Wan

2023Drug Discovery Today18 citationsDOI

Topics & Concepts

Drug discoveryDrugPharmacologyChemistryCytochrome P450Drug metabolismDrug reactionComputational biologyEnzymeMedicineBiochemistryBiologyPharmacogenetics and Drug MetabolismComputational Drug Discovery MethodsBiosimilars and Bioanalytical Methods
Preclinical evaluation of chemically reactive metabolites and mitigation of bioactivation in drug discovery | Litcius