Structural characterization of dicyanopyridine containing DNMT1-selective, non-nucleoside inhibitors
J.R. Horton, Sarath Pathuri, Kristen Wong, Ren Ren, Lourdes Rueda, David T. Fosbenner, Dirk A. Heerding, Michael T. McCabe, Melissa B. Pappalardi, Xing Zhang, Bryan W. King, Xiaodong Cheng
Topics & Concepts
DNA methylationDNACpG siteActive siteChemistryBiochemistryBiologyEpigeneticsEnzymeGeneGene expressionEpigenetics and DNA MethylationCancer-related gene regulationDNA and Nucleic Acid Chemistry