Litcius/Paper detail

Non-kinase off-target inhibitory activities of clinically-relevant kinase inhibitors

Nickolas R. Brauer, Allison L. Kempen, Delmis E. Hernandez, Herman O. Sintim

2024European Journal of Medicinal Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

KinomeKinaseDrug discoveryChemistryPharmacologyBiochemistryComputational biologyBiologyChronic Myeloid Leukemia TreatmentsHER2/EGFR in Cancer ResearchMelanoma and MAPK Pathways