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TGR5 agonist inhibits intestinal epithelial cell apoptosis via cAMP/PKA/c-FLIP/JNK signaling pathway and ameliorates dextran sulfate sodium-induced ulcerative colitis

Wenji Yang, Fanghui Han, Yipei Gu, Hui Qu, Jia Liu, Jianhua Shen, Ying Leng

2023Acta Pharmacologica Sinica47 citationsDOIOpen Access PDF

Topics & Concepts

ApoptosisSignal transductionColitisIntestinal epitheliumG protein-coupled bile acid receptorProtein kinase ACell biologyChemistryIntestinal mucosaKinasePharmacologyBiologyEndocrinologyReceptorInternal medicineImmunologyEpitheliumMedicineBiochemistryGeneticsDrug Transport and Resistance MechanismsBarrier Structure and Function StudiesPhagocytosis and Immune Regulation
TGR5 agonist inhibits intestinal epithelial cell apoptosis via cAMP/PKA/c-FLIP/JNK signaling pathway and ameliorates dextran sulfate sodium-induced ulcerative colitis | Litcius