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Exploration of chalcones as 3-chymotrypsin-like protease (3CLpro) inhibitors of SARS-CoV-2 using computational approaches

Thua-Phong Lam, Dac-Nhan Nguyen, Tan Thanh, Thanh‐Dao Tran, Minh-Tri Le, P. Huynh, Duc-Tuan Nguyen, Viet-Hung Tran, Dieu-Thuong Thi Trinh, Phuong Kim Truong, Cam‐Van T. Vo, Khac‐Minh Thai

2022Structural Chemistry13 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryIn silicoProteaseADMEDocking (animal)ChalconeStereochemistryEnzymeLigand (biochemistry)Molecular dynamicsBiochemistryIn vitroComputational chemistryCombinatorial chemistryReceptorGeneNursingMedicineComputational Drug Discovery MethodsSynthesis and biological activitythermodynamics and calorimetric analyses
Exploration of chalcones as 3-chymotrypsin-like protease (3CLpro) inhibitors of SARS-CoV-2 using computational approaches | Litcius