Design and synthesis of novel quinazolinyl-bisspirooxindoles as potent anti-tubercular agents: an ultrasound-promoted methodology
Bhargava Sai Allaka, Srinivas Basavoju, Estharla Madhu Rekha, Dharmarajan Sriram, Gamidi Rama Krishna
Topics & Concepts
Mycobacterium tuberculosisCytotoxicityCycloadditionChemistryDocking (animal)IC50Combinatorial chemistryMinimum inhibitory concentrationIn vitroStereochemistrySelectivitySonicationTuberculosisBiochemistryChromatographyMedicineCatalysisNursingPathologyQuinazolinone synthesis and applicationsSynthesis and biological activityMulticomponent Synthesis of Heterocycles