Piperazine-2-carboxylic acid derivatives as MTDLs anti-Alzheimer agents: Anticholinesterase activity, mechanistic aspect, and molecular modeling studies
Aya M. Soliman, Hend A. A. Abd El-wahab, Hülya Akıncıoğlu, İlhami Gülçın, Farghaly A. Omar
Topics & Concepts
ChemistryButyrylcholinesteraseAcetylcholinesteraseTacrinePiperazineAchéStereochemistryCarboxylic acidPharmacologyEnzymeBiochemistryOrganic chemistryMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity