Litcius/Paper detail

Development of phenyltriazole thiol-based derivatives as highly potent inhibitors of DCN1-UBC12 interaction

Wenjuan Zhou, Chenhao Xu, Guanjun Dong, Hui Qiao, Jing Yang, Hong‐Min Liu, Lina Ding, Kai Sun, Wen Zhao

2021European Journal of Medicinal Chemistry20 citationsDOIOpen Access PDF

Topics & Concepts

NeddylationChemistryCullinIC50Ubiquitin ligaseUbiquitinThiolIn vitroProtein–protein interactionBiochemistryGeneUbiquitin and proteasome pathwaysAutophagy in Disease and TherapyCancer-related Molecular Pathways