Fragment-based discovery of new potential DNMT1 inhibitors integrating multiple pharmacophore modeling, 3D-QSAR, virtual screening, molecular docking, ADME, and molecular dynamics simulation approaches
Goverdhan Lanka, Suvankar Banerjee, Nilanjan Adhikari, Balaram Ghosh
Topics & Concepts
PharmacophoreVirtual screeningADMEChemistryDocking (animal)Computational biologyEpigeneticsIn silicoQuantitative structure–activity relationshipSmall moleculeDrug discoveryStereochemistryDNMT1Combinatorial chemistryBiochemistryMethyltransferaseBiologyMethylationDNAIn vitroGeneMedicineNursingEpigenetics and DNA MethylationHIV/AIDS Research and InterventionsHIV/AIDS drug development and treatment