Fascaplysin derivatives binding to DNA via unique cationic five-ring coplanar backbone showed potent antimicrobial/antibiofilm activity against MRSA in vitro and in vivo
Xiao Wang, Hongda Qiu, Na Yang, Haoji Xie, Weida Liang, Jiayu Lin, Haifeng Zhu, Yuan Zhou, Ning Wang, Xinyi Tan, Zhou Jiale, Wei Cui, Da Teng, Jianhua Wang, Hongze Liang
Topics & Concepts
ChemistryCationic polymerizationAntimicrobialAntibacterial activityStaphylococcus aureusIn vivoIn vitroBiofilmCombinatorial chemistryAmideBacteriaStereochemistryBiochemistryOrganic chemistryBiologyBiotechnologyGeneticsSynthesis and bioactivity of alkaloidsAntimicrobial Peptides and ActivitiesBiochemical and Structural Characterization