Litcius/Paper detail

Fascaplysin derivatives binding to DNA via unique cationic five-ring coplanar backbone showed potent antimicrobial/antibiofilm activity against MRSA in vitro and in vivo

Xiao Wang, Hongda Qiu, Na Yang, Haoji Xie, Weida Liang, Jiayu Lin, Haifeng Zhu, Yuan Zhou, Ning Wang, Xinyi Tan, Zhou Jiale, Wei Cui, Da Teng, Jianhua Wang, Hongze Liang

2022European Journal of Medicinal Chemistry28 citationsDOI

Topics & Concepts

ChemistryCationic polymerizationAntimicrobialAntibacterial activityStaphylococcus aureusIn vivoIn vitroBiofilmCombinatorial chemistryAmideBacteriaStereochemistryBiochemistryOrganic chemistryBiologyBiotechnologyGeneticsSynthesis and bioactivity of alkaloidsAntimicrobial Peptides and ActivitiesBiochemical and Structural Characterization