Design and synthesis of novel 1,2,3-triazole linked hybrids: Molecular docking, MD simulation, and their antidiabetic efficacy as α-Amylase inhibitors
Ajayrajsinh R. Zala, Hem N. Naik, Iqrar Ahmad, Harun Patel, Smita Jauhari, Premlata Kumari
Topics & Concepts
ChemistryDocking (animal)In silicoActive siteEnzymeCoumarinTriazole1,2,3-TriazoleAmylaseIC50AcarboseStereochemistryBiochemistryIn vitroCombinatorial chemistryPharmacologyOrganic chemistryNursingMedicineGeneClick Chemistry and ApplicationsSynthesis and biological activityNatural Antidiabetic Agents Studies