Discovery of spirooxadiazoline oxindoles with dual-stage antimalarial activity
Elizabeth A. Lopes, Raquel Mestre, Diana Fontinha, Jenny Legac, Jinxin V. Pei, Margarida Sanches‐Vaz, Mattia Mori, Adele M. Lehane, Philip J. Rosenthal, Miguel Prudêncio, Maria M. M. Santos
Topics & Concepts
MalariaPlasmodium falciparumPlasmodium bergheiChemistryArtemisininPharmacologyAntimalarial AgentMechanism of actionEffluxDrug discoveryIn vitroBiochemistryBiologyImmunologyMalaria Research and ControlTrypanosoma species research and implicationsHIV/AIDS drug development and treatment