Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers
Tithi Roy, Samuel Boateng, Sergette Banang‐Mbeumi, Pankaj Kumar Singh, Pratik Basnet, Roxane-Cherille N. Chamcheu, Federico Ladu, Isabel M. Chauvin, Vladimir S. Spiegelman, Ronald A. Hill, Konstantin G. Kousoulas, Bolni Marius Nagalo, Anthony L. Walker, Jean Fotie, Siva Murru, Mario Sechi, Jean Christopher Chamcheu
Topics & Concepts
FisetinPI3K/AKT/mTOR pathwayKinasePharmacologyDocking (animal)ChemistryCancer researchMelanomaBiochemistryApoptosisBiologyQuercetinMedicineNursingAntioxidantFlavonoids in Medical ResearchBiological Activity of Diterpenoids and BiflavonoidsFungal Biology and Applications