Litcius/Paper detail

Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers

Tithi Roy, Samuel Boateng, Sergette Banang‐Mbeumi, Pankaj Kumar Singh, Pratik Basnet, Roxane-Cherille N. Chamcheu, Federico Ladu, Isabel M. Chauvin, Vladimir S. Spiegelman, Ronald A. Hill, Konstantin G. Kousoulas, Bolni Marius Nagalo, Anthony L. Walker, Jean Fotie, Siva Murru, Mario Sechi, Jean Christopher Chamcheu

2020Bioorganic Chemistry34 citationsDOIOpen Access PDF

Topics & Concepts

FisetinPI3K/AKT/mTOR pathwayKinasePharmacologyDocking (animal)ChemistryCancer researchMelanomaBiochemistryApoptosisBiologyQuercetinMedicineNursingAntioxidantFlavonoids in Medical ResearchBiological Activity of Diterpenoids and BiflavonoidsFungal Biology and Applications