Discovery of quinazolinyl-containing benzamides derivatives as novel HDAC1 inhibitors with in vitro and in vivo antitumor activities
Zixue Zhang, Qingwei Zhang, Hao Zhang, Min-Ru Jiao, Zheng Guo, Xinyan Peng, Lei Fu, Jianqi Li
Topics & Concepts
ChemistryHDAC1HDAC8BenzamideIn vivoIn vitroHistone deacetylaseHDAC6PharmacologyHistone deacetylase 2Cancer researchBiochemistryHistoneStereochemistryBiologyBiotechnologyGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis