Design, synthesis, and biological evaluation of novel imidazole derivatives possessing terminal sulphonamides as potential BRAFV600Einhibitors
Eslam M.H. Ali, Mohammed S. Abdel‐Maksoud, Usama M. Ammar, Karim I. Mersal, Kyung Ho Yoo, Park Jooryeong, Chang‐Hyun Oh
Topics & Concepts
ChemistryIC50Cancer cell linesCell cultureImidazoleMelanomaCombinatorial chemistryCancerKinaseCancer cellLead compoundStereochemistryIn vitroCancer researchBiochemistryBiologyInternal medicineMedicineGeneticsMelanoma and MAPK PathwaysComputational Drug Discovery MethodsSynthesis and biological activity