First-in-human phase I study of JPH203, an L-type amino acid transporter 1 inhibitor, in patients with advanced solid tumors
Naohiro Okano, Daisuke Naruge, Kirio Kawai, Takaaki Kobayashi, Fumio Nagashima, Hitoshi Endou, Junji Furuse
Topics & Concepts
MedicineGastroenterologyInternal medicinePharmacokineticsN-acetyltransferaseResponse Evaluation Criteria in Solid TumorsPharmacologyDiseaseProgressive diseaseChemistryGeneBiochemistryAcetylationAmino Acid Enzymes and MetabolismEpigenetics and DNA MethylationDrug Transport and Resistance Mechanisms