Chrysin based pyrimidine-piperazine hybrids: design, synthesis, in vitro antimicrobial and in silico E. coli topoisomerase II DNA gyrase efficacy
Kajalben B. Patel, Dhanji P. Rajani, Iqrar Ahmad, Harun Patel, Hitesh D. Patel, Premlata Kumari
Topics & Concepts
DNA gyraseNorfloxacinAntimicrobialChemistryProtein Data Bank (RCSB PDB)PiperazineTopoisomerase IVDocking (animal)Candida albicansBiochemistryBiologyEscherichia coliMicrobiologyCiprofloxacinPharmacologyAntibioticsMedicineNursingGeneCancer therapeutics and mechanismsBioactive Compounds and Antitumor AgentsSynthesis and biological activity