Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson’s Disease
Rita Maria Concetta Di Martino, Letizia Pruccoli, Alessandra Bisi, Silvia Gobbi, Angela Rampa, Ana Martı́nez, Concepción Pérez, Loreto Martínez‐González, Maria Paglione, Elia Di Schiavi, Francesca Seghetti, Andrea Tarozzi, Federica Belluti
Abstract
emerged as an interesting multitarget derivative, valuable to be exploited in a multitarget PD perspective.
Topics & Concepts
NeuroprotectionCurcuminNeurotoxicityOxidative stressNeuroinflammationPharmacologyParkinson's diseaseAntioxidantInducerChemistryDownregulation and upregulationBiologyNeuroscienceBiochemistryMedicineDiseaseInternal medicineToxicityGeneOrganic chemistryGenomics, phytochemicals, and oxidative stressCurcumin's Biomedical ApplicationsCholinesterase and Neurodegenerative Diseases