Piperidine-4-carboxamide as a new scaffold for designing secretory glutaminyl cyclase inhibitors
K.V. Dileep, Naoki Sakai, Kentaro Ihara, M. Kato-Murayama, Akiko Nakata, Akihiro Ito, Divya M. Sivaraman, Jay W. Shin, Minoru Yoshida, Mikako Shirouzu, Kam Y. J. Zhang
Topics & Concepts
Virtual screeningPharmacophorePiperidineMoietyDocking (animal)CarboxamideChemistryCyclasePharmacologyComputational biologyBiochemistryEnzymeMedicineBiologyStereochemistryNursingAlzheimer's disease research and treatmentsAmino Acid Enzymes and MetabolismDrug Transport and Resistance Mechanisms