Identification of novel ureido benzothiophenes as dual VEGFR-2/EGFR anticancer agents
Wagdy M. Eldehna, Ghada H. Al-Ansary, Tarfah Al‐Warhi, Maiy Y. Jaballah, Mahmoud M. Elaasser, Mahmoud Rashed
Topics & Concepts
ChemistryErlotinibCytotoxic T cellIC50SorafenibKinaseBenzothiopheneStereochemistryThioureaEGFR inhibitorsThiopheneCancer researchPharmacologyBiochemistryEpidermal growth factor receptorIn vitroReceptorOrganic chemistryHepatocellular carcinomaMedicineBiologyCancer, Hypoxia, and MetabolismSynthesis and biological activityPI3K/AKT/mTOR signaling in cancer