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Evybactin is a DNA gyrase inhibitor that selectively kills Mycobacterium tuberculosis

Yu Imai, Glenn Hauk, Jeffrey Quigley, Libang Liang, Sangkeun Son, Meghan Ghiglieri, Michael F. Gates, Madeleine Morrissette, Negar Shahsavari, Samantha Niles, Donna M. Baldisseri, Chandrashekhar Honrao, Xiaoyu Ma, Jason J. Guo, James M. Berger, Kim Lewis

2022Nature Chemical Biology61 citationsDOIOpen Access PDF

Topics & Concepts

DNA gyraseMycobacterium tuberculosisMicrobiologyAntibioticsAntimicrobialTuberculosisBiologyAntibiotic resistanceMycobacteriumNovobiocinChemistryComputational biologyBacteriaGeneticsGeneMedicineEscherichia coliPathologyCancer therapeutics and mechanismsAntibiotic Resistance in BacteriaMicrobial Natural Products and Biosynthesis
Evybactin is a DNA gyrase inhibitor that selectively kills Mycobacterium tuberculosis | Litcius