Novel orally bioavailable piperidine derivatives as extracellular arginase inhibitors developed by a ring expansion
Anna Gzik, Bartłomiej Borek, Jacek Chrzanowski, Karol Jedrzejczak, Marek Dzięgielewski, Joanna Brzezińska, Julita Nowicka, Marcin Grzybowski, Tomasz Rejczak, Dorota Niedziałek, Grzegorz Wieczorek, Jacek Olczak, Adam Gołȩbiowski, Zbigniew Zasłona, Roman Błaszczyk
Topics & Concepts
ChemistryArginaseBioavailabilityPharmacologyIn vivoBiochemistryAmino acidMedicineBiologyArginineBiotechnologyPneumocystis jirovecii pneumonia detection and treatmentAmino Acid Enzymes and MetabolismSynthesis and Catalytic Reactions