Development of inhibitors targeting glycogen synthase kinase-3β for human diseases: Strategies to improve selectivity
Junxia Wei, Jiaxing Wang, Jifa Zhang, Jinliang Yang, Guan Wang, Yuxi Wang
Topics & Concepts
GSK-3ChemistryGlycogen synthaseKinaseThreonineSerineEnzymeSelectivityGSK3BBiochemistrySignal transductionPharmacologyBiologyCatalysisWnt/β-catenin signaling in development and cancerCancer-related gene regulationProtein Degradation and Inhibitors